Product Specifications Research Overview Melanotan I, also written Melanotan 1 or MT1, is the linear tridecapeptide [Nle, D-Phe]-alpha-melanocyte-stimulating hormone, catalogued in the literature as afamelanotide and as NDP-alpha-MSH, sequence Ac-Ser-Tyr-Ser-Nle-Glu-His-D-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH (CHNO, 1646.9 g/mol, CAS 75921-69-6)
Biased Agonism and -Opioid Receptor Regulation The literature contains numerous examples of agonist-selective regulation of opioid receptors and this has been reviewed previously (Koch and Hlt, 2008

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